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I-Micafungin ye-antifungal kanye ne-antiviral

Incazelo emfushane:

Igama: Micafungin

Inombolo ye-CAS: 235114-32-6

Ifomula yemolekyuli: C56H71N9O23S

Isisindo se-molecule: 1270.28

Inombolo ye-EINECS: 1806241-263-5


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Imininingwane Yomkhiqizo

Igama I-Micafungin
Inombolo ye-CAS 235114-32-6
Ifomula yamangqamuzana I-C56H71N9O23S
Isisindo samangqamuzana 1270.28
Inombolo ye-EINECS 1806241-263-5

I-Clinical Pharmacology

Lo mkhiqizo owokujova nge-intravenous.Ukuhlushwa kwe-plasma kufinyelela kumkhawulo ekugcineni kokumnika, kanti isigamu sempilo singamahora ayi-13.9.Ukugcwala kwe-micafungin emaphashini, esibindini, ubendeni nasezicutshini zezinso kuphezulu kakhulu, kodwa akutholakali oketshezini lwe-cerebrospinal.Ngemuva kokujova nge-intravenous, ikakhulukazi i-metabolized esibindini futhi ikhishwe indle nomchamo.

Umsebenzi

Umthamo onconyiwe wokwelashwa kwe-candidiasis esophageal ngu-150 mg ngosuku, futhi umthamo onconyiwe wokuvikela ukutheleleka kwe-Candida ezigulini zokufakelwa kwe-hematopoietic stem cell ngu-50 mg ngosuku.Ngokusho kwedatha yomtholampilo etholakalayo, inkambo evamile yokwelashwa noma ukuvimbela izifo ezimbili ezingenhla yizinsuku ezingu-15 nezinsuku ezingu-19, ngokulandelana.Umuthi ulungiswa futhi uhlanjululwe ngomjovo we-saline ojwayelekile noma umjovo we-dextrose ongu-5%.Isikhathi sokuphatha kufanele sibe okungenani ihora elingu-1, ngaphandle kwalokho kulula ukukhiqiza ukusabela okubi.

Ukusebenzisana Kwemithi

Izinga eliphakeme le-plasma ye-nifedipine lingakhuphuka ngo-42%, futhi uma kunesidingo, cabanga ukunciphisa umthamo we-nifedipine noma ukuyeka umuthi.Indawo engaphansi kwejika lokuhlushwa le-plasma lomuthi olwa nokwenqaba isitho iSirolimus inyuke ngo-21%, futhi ukuncipha komthamo we-sirolimus kufanele kubhekwe njengokufanelekile.Izidakamizwa ze-antifungal, i-pharmacology yomtholampilo, ukusetshenziswa, ukusabela okubi, njll. ye-micafungin

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