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I-Tirzepatide Powder Yomjovo Wokunciphisa Isisindo 30mg Nge-Vial Purity 99%

Incazelo emfushane:

Igama: I-Tirzepatide Injection Powder

Ubumsulwa: 99%

Usayizi: 30mg

Amanzi: 3.0%

Ukubukeka: I-White Lyophilized Powder

Ukunyibilika: Kuyavumelana

Ukuqinisekiswa kwe-HPLC: Kuyavumelana

Ama-Endotoxin Amagciwane: Ngaphansi kwe-5 EU/mg

Ukuqinisekiswa kwe-MS: 4810.6

Izinzuzo: Ukunciphisa Isisindo


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Incazelo

I-Tirzepatide iyinoveli, i-insulinotropic polypeptide (GIP) esebenza kabili esebenza ngeglucose ne-glucagon-like peptide-1 (GLP-1) receptor agonist. Imele intuthuko enkulu ekwelapheni uhlobo lwesifo sikashukela sohlobo 2 futhi ibonise imiphumela ethembisayo ekulawuleni isisindo. I-Tirzepatide injection powder iyifomu lezemithi elisetshenziselwa ukulungisa isisombululo sokuphathwa kwe-subcutaneous.

Indlela Yokwenza
I-Tirzepatide isebenza ngokwenza kokubili ama-receptors e-GIP kanye ne-GLP-1, abambe iqhaza ekulawuleni amazinga kashukela egazini kanye nesifiso sokudla. I-agonism emibili inikeza imiphumela eminingi enenzuzo:

Ukukhiqizwa Kwe-insulin Okuthuthukisiwe: Ivuselela ukukhishwa kwe-insulin ngendlela encike kushukela, isiza ukwehlisa amazinga kashukela ngaphandle kokubanga i-hypoglycemia.
Ukukhishwa Kwe-Glucagon Ecindezelwe: Yehlisa ukukhiqizwa kwe-glucagon, i-hormone enyusa amazinga kashukela egazini.
I-Appetite Regulation: Ikhuthaza ukusutha futhi inciphisa ukudla, okunomthelela ekwehleni kwesisindo.
I-Slowed Gastric Emptying: Ibambezela ukuphuma kwesisu, okusiza ekulawuleni ukukhuphuka koshukela wegazi ngemuva kokudla.

Ukusetshenziswa Okugunyaziwe
Njengezibuyekezo zakamuva, i-Tirzepatide igunyazwe iziphathimandla ezilawulayo ezifana ne-US Food and Drug Administration (FDA) yokwelashwa kohlobo 2 lwesifo sikashukela. Iphinde iphenywe ngokusetshenziswa kwayo ekulawulweni kokukhuluphala.

Izinzuzo
Ukulawula I-Glycemic Okusebenzayo: Ukuncipha okukhulu kumazinga e-HbA1c.
Ukunciphisa Isisindo: Ukunciphisa isisindo esikhulu, okuwusizo ezigulini ezinesifo sikashukela sohlobo 2 kanye nokukhuluphala.
Izinzuzo zenhliziyo nemithambo yegazi: Intuthuko engaba khona ezicini eziyingozi zenhliziyo, nakuba izifundo eziqhubekayo zisahlola lesi sici.
Ukunethezeka: Umthamo kanye ngeviki uthuthukisa ukubambelela kwesiguli uma kuqhathaniswa nemithi yansuku zonke.

Engase Engase Side Effects
Nakuba i-Tirzepatide ivame ukubekezelelwa kahle, abanye abasebenzisi bangase babe nemiphumela emibi, kuhlanganise:

Izinkinga zeGastrointestinal:

Isicanucanu, ukuhlanza, isifo sohudo, nokuqunjelwa kuvamile, ikakhulukazi phakathi nezigaba zokuqala zokwelashwa.
Ingozi ye-Hypoglycemia: Ikakhulukazi uma isetshenziswa ngokuhlangana neminye imithi yokwehlisa ushukela.
I-Pancreatitis: Okungavamile kodwa kubi kakhulu, okudinga ukunakekelwa ngokushesha uma kuvela izimpawu ezinjengobuhlungu besisu obukhulu.

Ukulungiselela Nokuphatha
I-Tirzepatide injection powder idinga ukuphinda ihlanganiswe ne-solvent efanelekile (evame ukunikezwa kukhithi) ukwenza isisombululo sokujova. Isixazululo esihlanganisiwe kufanele sicace futhi singabi nezinhlayiya. Ilawulwa ngaphansi kwesikhumba esiswini, ethangeni, noma engalweni engenhla.


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