Ukunamathela enkolelweni "Yokudala izinto ezisezingeni eliphezulu nokudala ubungane nabantu namuhla abavela emhlabeni wonke", sivame ukubeka isithakazelo sabathengi endaweni yokuqala ngentengo ecashuniwe ye-China Healthy Weight Loss CAS 96829-58-2 99% Bulk API Rimonbant CetilistatI-Orlistat, Kusukela sasungulwa ekuqaleni kwawo-1990, manje sesakhe inethiwekhi yethu yokuthengisa e-USA, Germany, Asia, kanye namazwe amaningana aseMpumalanga Ephakathi. Sihlose ukuthola umphakeli wezinga eliphezulu emhlabeni wonke we-OEM kanye ne-aftermarket!
Ukunamathela enkolelweni "Yokudala izinto ezisezingeni eliphezulu nokudala ubungane nabantu namuhla abavela kuwo wonke umhlaba", sivame ukubeka izithakazelo zabathengi kuqalaI-China 96829-58-2, I-Orlistat, Ngohlelo olusezingeni eliphezulu lokumaketha oluphelele kanye nokuzikhandla kwabasebenzi abangu-300 abanamakhono, inkampani yethu ithuthukise zonke izinhlobo zezixazululo ezisukela ekilasini eliphezulu, eliphakathi kuya esigabeni esiphansi. Lonke lolu khetho lwezinto ezinhle lunikeza amakhasimende ethu ukukhetha okuhlukile. Ngaphandle kwalokho, inkampani yethu inamathela kukhwalithi ephezulu namanani aphusile, futhi sikunikeza nezinsizakalo ezinhle ze-OEM ezinkampanini eziningi ezidumile.
| Igama | I-Leuprorelin |
| Inombolo ye-CAS | 53714-56-0 |
| Ifomula yamangqamuzana | I-C59H84N16O12 |
| Isisindo samangqamuzana | 1209.4 |
| Inombolo ye-EINECS | 633-395-9 |
| Ukuzungezisa okuqondile | I-D25 -31.7° (c = 1 ku-1% i-acetic acid) |
| Ukuminyana | 1.44±0.1 g/cm3(Kubikezelwe) |
| Isimo sesitoreji | -15°C |
| Ifomu | Icocekile |
| I-acidity coefficient | (pKa) 9.82±0.15 (Kubikezelwe) |
| Ukuncibilika kwamanzi | Incibilika emanzini ngo-1mg/ml |
LH-RHLEUPROLIDE;LEUPROLIDE;LEUPROLIDE(HUMAN);LEUPRORELIN;[DES-GLY10,D-LEU6,PRO-NHET9]-LUTEINIZINGHORMONE-RELEASINGHORMONEHUMAN;(DES-GLY10,D-LEU6,PRO -NHET9)-LUTEINIZINGHORMONE-RELEASINGHORMONE;(DES-GLY10,D-LEU6,PRO-NHET9)-LUTEINIZINGHORMONE-REASINGIFACTOR;[DES-GLY10,D-LEU6,PRO-NHET9]-LH-RH(HUMAN)
I-Leuprolide, i-goserelin, i-triprelin, ne-nafarelin yizidakamizwa ezimbalwa ezivame ukusetshenziswa emtholampilo ukuze kukhishwe ama-ovari ukuze kwelashwe umdlavuza webele wangaphambi kokuya esikhathini kanye nomdlavuza wendlala yesinye. (okubizwa ngokuthi izidakamizwa ze-GnRH-a), izidakamizwa ze-GnRH-a ziyafana ngesakhiwo se-GnRH futhi zincintisana nama-pituitary GnRH receptors. Okusho ukuthi, i-gonadotropin ekhiqizwe yi-pituitary iyancipha, okuholela ekwehleni okukhulu kwehomoni yocansi ekhishwa i-ovary.
I-Leuprolide iyi-analog ye-gonadotropin-releasing hormone (GnRH), i-peptide eyakhiwe ngama-amino acid ayi-9. Lo mkhiqizo ungavimbela ngokuphumelelayo ukusebenza kwesistimu ye-pituitary-gonadal, ukumelana nama-enzyme e-proteolytic kanye nokuhlobana ne-pituitary GnRH receptor kunamandla kune-GnRH, futhi umsebenzi wokugqugquzela ukukhululwa kwe-hormone ye-luteinizing (LH) cishe izikhathi ezingu-20 kune-GnRH. Iphinde ibe nomthelela onamandla ovimbelayo ekusebenzeni kwe-pituitary-gonad kune-GnRH. Esigabeni sokuqala sokwelashwa, i-follicle stimulating hormone (FSH), LH, estrogen noma i-androgen ingase ikhule okwesikhashana, bese kuthi, ngenxa yokuncipha kokusabela kwe-pituitary gland, ukukhishwa kwe-FSH, LH ne-estrogen noma i-androgen kuvinjelwe, okuholela ekuthembeleni kumahomoni ocansi. Izifo zocansi (ezifana nomdlavuza wendlala yesinye, i-endometriosis, njll.) zinomphumela wokwelapha.
Njengamanje, usawoti we-acetate we-leuprolide usetshenziswa kakhulu emtholampilo, ngoba ukusebenza kwe-leuprolide acetate kuzinzile ekamelweni lokushisa. Uketshezi kufanele kulahlwe. Ingasetshenziselwa ukwelashwa kokuthenwa kwezidakamizwa kwe-endometriosis kanye ne-uterine fibroids, ukuthomba okuphakathi, umdlavuza webele we-premenopausal kanye nomdlavuza wendlala yesinye, kanye nokopha okusebenzayo kwesibeletho okuphikisiwe noma okungasebenzi ekwelapheni okujwayelekile kwama-hormone. Ingasetshenziswa futhi njengomuthi wokwelapha ngaphambi kokukhishwa kwe-endometrial, okunganciphisa i-endometrium ngokulinganayo, kwehlise i-edema, futhi kunciphise nobunzima bokuhlinzwa. Ukunamathela enkolelweni “Yokudala izinto ezisezingeni eliphezulu nokudala ubungane nabantu namuhla abavela kuwo wonke umhlaba”, ngokuvamile sibeka isithakazelo sabathengi kuqala ngentengo ecashuniwe ye-China Healthy 92 Isisindo 92 Isisindo 92 Isisindo Sokukhulu 92 Isisindo 92 Isisindo 98 I-API Rimonbant Cetilistat Orlistat, Kusukela yasungulwa ekuqaleni kwawo-1990, manje sesakhe inethiwekhi yethu yokuthengisa e-USA, Germany, Asia, kanye namazwe amaningana aseMpumalanga Ephakathi. Sihlose ukuthola umphakeli wezinga eliphezulu emhlabeni wonke we-OEM kanye ne-aftermarket!
Intengo ecashuniwe yeI-China 96829-58-2, I-Orlistat, Ngohlelo lwempendulo yokuthengisa olusezingeni eliphezulu kanye nokusebenza kanzima kwabasebenzi abangu-300 abanamakhono, inkampani yethu ithuthukise zonke izinhlobo zezixazululo kusukela kusigaba esiphakeme, esiphakathi kuya esigabeni esiphansi. Lonke lolu khetho lwezinto ezinhle lunikeza amakhasimende ethu ukukhetha okuhlukile. Ngaphandle kwalokho, inkampani yethu inamathela kukhwalithi ephezulu namanani aphusile, futhi sikunikeza nezinsizakalo ezinhle ze-OEM ezinkampanini eziningi ezidumile.