Peptide APIs
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NMN
Ucwaningo lwangaphambi komtholampilo kanye nolwasekuqaleni kwabantu luphakamisa ukuthi i-NMN ingase ikhuthaze ukuphila isikhathi eside, ukukhuthazela ngokomzimba, nokusebenza kwengqondo.
Izici ze-API:
Ukuhlanzeka okuphezulu ≥99%
Ibanga lezemithi, elilungele ukwakheka ngomlomo noma okujovwayo
Kwenziwe ngaphansi kwamazinga afana ne-GMP
I-NMN API ilungele ukusetshenziswa ezithasiselweni zokulwa nokuguga, ukwelashwa kwe-metabolic, kanye nocwaningo lwempilo ende.
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IGlucagon
I-Glucagon iyi-hormone yemvelo ye-peptide esetshenziswa njengokwelashwa okuphuthumayo kwe-hypoglycemia enzima futhi yafundelwa indima yayo ekulawuleni i-metabolic, ukuncipha kwesisindo, kanye nokuxilongwa kokugaya ukudla.
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I-Motixafortide
I-Motixafortide iyi-peptide yokwenziwa ye-CXCR4 ephikisanayo eyenzelwe ukuhlanganisa amangqamuzana e-hematopoietic stem (HSCs) ukuze kufakwe i-autologous transplantation futhi iyacwaningwa ku-oncology kanye ne-immunotherapy.
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I-Glepaglutide
I-Glepaglutide iyi-analog esebenza isikhathi eside ye-GLP-2 eyenzelwe ukwelapha i-short bowel syndrome (SBS). Ithuthukisa ukumuncwa nokukhula kwamathumbu, kusize iziguli zehlise ukuncika ekondlekeni kwabazali.
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I-Elamipretide
I-Elamipretide iyi-tetrapeptide ehloselwe i-mitochondria eyenzelwe ukwelapha izifo ezibangelwa ukungasebenzi kahle kwe-mitochondrial, okuhlanganisa i-mitochondrial myopathy eyinhloko, i-Barth syndrome, nokuhluleka kwenhliziyo.
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I-Pegcetacoplan
I-Pegcetacoplan iyipeptide ye-pegylated cyclic esebenza njenge-C3 complement inhibitor ehlosiwe, eyenzelwe ukwelashwa kwezifo ezihambisanayo ezifana ne-paroxysmal nocturnal hemoglobinuria (PNH) kanye ne-geographic atrophy (GA) ekuwohlokeni kwe-macular okuhlobene neminyaka.
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I-Palopegteriparatide
I-Palopegteriparatide iyi-agonist esebenza isikhathi eside ye-parathyroid hormone receptor (PTH1R agonist), eyenzelwe ukwelashwa kwe-hypoparathyroidism engapheli. Kuyi-analog ye-pegylated ye-PTH (1-34) eklanyelwe ukunikeza ukulawulwa kwe-calcium okuqhubekayo ngokudosa kanye ngeviki.
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I-GHRP-6
I-GHRP-6 (I-Growth Hormone Releasing Peptide-6) iyi-hexapeptide yokwenziwa esebenza njenge-secretagogue ye-hormone yokukhula, evuselela ukukhululwa kwemvelo komzimba kwe-hormone yokukhula (GH) ngokwenza kusebenze isamukeli se-GHSR-1a.
Izici ze-API :
Ukuhlanzeka ≥99%
Kwenziwe nge-solid-phase peptide synthesis (SPPS)
Ihlinzekelwe i-R&D nokusetshenziswa kwezentengiso
I-GHRP-6 iyi-peptide yocwaningo enemisebenzi eminingi yokusekelwa kwe-metabolic, ukuvuselelwa kwemisipha, nokuguqulwa kwamahomoni.
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I-GHRP-2
I-GHRP-2 (I-Growth Hormone Releasing Peptide-2) iyi-hexapeptide yokwenziwa kanye ne-hormone yokukhula enamandla secretagogue, eklanyelwe ukugqugquzela ukukhululwa kwemvelo kwe-hormone yokukhula (GH) ngokwenza kusebenze isamukeli se-GHSR-1a ku-hypothalamus kanye ne-pituitary.
Izici ze-API:
Ukuhlanzeka ≥99%
Itholakalela i-R&D kanye nokuhlinzekwa kwezentengiso, nemibhalo egcwele ye-QC
I-GHRP-2 iyi-peptide yocwaningo ebalulekile emikhakheni ye-endocrinology, imithi evuselelayo, kanye nokwelashwa okuhlobene nobudala.
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I-Hexarelin
I-Hexarelin iyi-hormone yokukhula yokwenziwa ye-secretagogue peptide (GHS) kanye ne-GHSR-1a agonist enamandla, ethuthukiswe ukugqugquzela ukukhululwa kwe-endogenous growth hormone (GH). Ingokomndeni we-ghrelin mimetic futhi yakhiwe ama-amino acid ayisithupha (i-hexapeptide), enikeza ukuzinza okuthuthukisiwe kwe-metabolic kanye nemiphumela eqinile yokukhulula i-GH uma kuqhathaniswa nama-analog angaphambilini afana ne-GHRP-6.
Izici ze-API :
Ukuhlanzeka ≥ 99%
Ikhiqizwe nge-solid-phase peptide synthesis (SPPS)
Amazinga afana ne-GMP, i-endotoxin ephansi nezinsalela ze-solvent
Ukunikezwa okuguquguqukayo: I-R&D kuya esikalini sezentengiso
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I-Melanotan II
Izici ze-API:
Ukuhlanzeka okuphezulu ≥ 99%
Ihlanganiswe nge-solid-phase peptide synthesis (SPPS)
I-endotoxin ephansi, izincibilikisi eziyinsalela ephansi
Itholakala nge-R&D kuya esikalini sezentengiso -
I-Melanotan 1
I-Melanotan 1 API ikhiqizwa kusetshenziswa ubuchwepheshe obuqinile besigaba se-peptide synthesis (SPPS) ngaphansi kwezimo eziqinile zokulawula ikhwalithi ezifana ne-GMP.
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Ukuhlanzeka okuphezulu ≥99%
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I-Solid-phase peptide synthesis (SPPS)
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Amazinga okukhiqiza afana ne-GMP
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Imibhalo egcwele: COA, MSDS, idatha yokuzinza
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Ukunikezwa okulinganiswayo: I-R&D kuya kumaleveli ezohwebo
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