I-Melanotan 1iyi-analog ye-peptide yokwenziwaI-α-MSH (i-alpha-melanocyte stimulating hormone). Isebenza ngeisebenze i-melanocortin-1 receptors (MC1R)ukugqugquzelaukukhiqizwa kwe-melanin, ukunikela ngemveloisikhumba sombalafuthiukuvikela isithombe.
Sekuyikugunyazwe ukwelashwa kwe-erythropoietic protoporphyria (EPP)-ukuphazamiseka okungajwayelekile okubangela ukuzwela okukhulu ekukhanyeni kwelanga. I-Melanotan 1 isiza ukwandaukubekezelela ukukhanya kwe-UV, nciphisaukusabela kwe-phototoxic, futhi uthuthukiseukuvikela isikhumba emonakalweni we-UV.
UkukhethaI-MC1R i-agonist
Iyakhulaukukhiqizwa kwe-eumelanin
Ihlinzekaukuvikelwa kwelanga kwemvelo
IsekelaUkulungiswa kwe-DNA kanye nempendulo elwa nokuvuvukala
Amathuba okuthii-vitiligo, ukuvimbela umdlavuza wesikhumba, futhii-cosmetic pigmentation
Kuhlolwe ngaphakathianti-ukugugafuthiukwelashwa kwe-dermatological
Ukuhlanzeka okuphezulu ≥99%
I-Solid-phase peptide synthesis (SPPS)
Amazinga okukhiqiza afana ne-GMP
Ukunikezwa okulinganiswayo: I-R&D kuya kumaleveli ezohwebo